Article Figures & Data
Figures
- FIGURE 1.
Synthetic schemes of click reactions: CuAAC (A), SPAAC (B), Diels-Alder reaction (C), and Staudinger ligation (D), and 2 variations on click-to-chelate radiolabeling methodology using CuAAC and 99mTc(CO)3 (E).
- FIGURE 2.
(A) Synthesis of 18F-RGD-K5. (B) Decay-corrected anterior maximum-intensity PET projections of female volunteer injected with 18F-RGD-K5.
- FIGURE 3.
(A) Synthetic route to 18F-transcyclooctene. (B) Synthesis of PARP1 inhibitor 18F-AAZD2281 using inverse electron-demand Diels-Alder click chemistry. (C) Schematic for methodology for pretargeted 64Cu-immunoPET imaging agent based on inverse electron Diels-Alder click chemistry. TCO = transcyclooctene.
