GRP receptor-targeted PET of a rat pancreas carcinoma xenograft in nude mice with a 68Ga-labeled bombesin (6–14) analog

J Schuhmacher, H Zhang, J Doll… - Journal of nuclear …, 2005 - Soc Nuclear Med
Bombesin (BN), a 14-amino-acid peptide, shows high affinity for the human gastrin-
releasing peptide receptor (GRP-r), which is overexpressed on several types of cancer …

PET of tumors expressing gastrin-releasing peptide receptor with an 18F-labeled bombesin analog

I Dijkgraaf, GM Franssen, WJ McBride… - Journal of Nuclear …, 2012 - Soc Nuclear Med
The gastrin-releasing peptide receptor (GRPR) is overexpressed in human prostate cancer.
Bombesin (BBN) is a neurotransmitter of 14 amino acids and binds with selectivity and with …

18F-labeled bombesin analogs for targeting GRP receptor-expressing prostate cancer

X Zhang, W Cai, F Cao, E Schreibmann… - Journal of Nuclear …, 2006 - Soc Nuclear Med
The gastrin-releasing peptide receptor (GRPR) is found to be overexpressed in a variety of
human tumors. The aim of this study was to develop 18F-labeled bombesin analogs for PET …

Bombesin antagonist–based radioligands for translational nuclear imaging of gastrin-releasing peptide receptor–positive tumors

K Abiraj, R Mansi, ML Tamma, M Fani… - Journal of Nuclear …, 2011 - Soc Nuclear Med
Bombesin receptors are overexpressed on a variety of human tumors. In particular, the
gastrin-releasing peptide receptor (GRPr) has been identified on prostate and breast …

18F-labeled bombesin analog for specific and effective targeting of prostate tumors expressing gastrin-releasing peptide receptors

M Honer, L Mu, T Stellfeld, K Graham… - Journal of Nuclear …, 2011 - Soc Nuclear Med
Bombesin is a peptide exhibiting high affinity for the gastrin-releasing peptide receptor
(GRPr), which is highly overexpressed on prostate cancer cells. In the present study, we …

Synthesis and radiopharmacological evaluation of a high-affinity and metabolically stabilized 18F-labeled bombesin analogue for molecular imaging of gastrin …

S Richter, M Wuest, SS Krieger, BE Rogers… - Nuclear Medicine and …, 2013 - Elsevier
Abstract Introduction Bombesin (BBN) and BBN analogues have attracted much attention as
high-affinity ligands for selective targeting of the gastrin-releasing peptide (GRP) receptor …

GRPR-selective PET imaging of prostate cancer using [18F]-lanthionine-bombesin analogs

G Carlucci, A Kuipers, HJK Ananias, D de Paula Faria… - Peptides, 2015 - Elsevier
The gastrin-releasing peptide receptor (GRPR) is overexpressed in a variety of human
malignancies, including prostate cancer. Bombesin (BBN) is a 14 amino acids peptide that …

Bombesin analogues for gastrin-releasing peptide receptor imaging

PK Nanda, U Pandey, BN Bottenus, TL Rold… - Nuclear medicine and …, 2012 - Elsevier
OBJECTIVES: The present study describes the design and development of a series of new
bombesin (BBN) antagonist peptide ligands of the form [64Cu-(NO2A-XD-Phe6-BBN (6-13) …

A comparative study of radiolabeled bombesin analogs for the PET imaging of prostate cancer

Y Liu, X Hu, H Liu, L Bu, X Ma, K Cheng… - Journal of nuclear …, 2013 - Soc Nuclear Med
Radiolabeled bombesin (BBN) analogs that bind to the gastrin-releasing peptide receptor
(GRPR) represent a topic of active investigation for the development of molecular probes for …

MicroPET Imaging of a Gastrin-Releasing Peptide Receptor-Positive Tumor in a Mouse Model of Human Prostate Cancer Using a 64Cu-Labeled Bombesin Analogue

BE Rogers, HM Bigott, DW McCarthy… - Bioconjugate …, 2003 - ACS Publications
The gastrin-releasing peptide receptor (GRPR) is overexpressed on a variety of carcinomas
and has been the target for detection and treatment of these neoplasms in animals. In …