Technetium-99m-labeled HOE 140: a potential bradykinin B2 receptor imaging agent

J Med Chem. 1995 Jul 21;38(15):2799-801. doi: 10.1021/jm00015a001.
No abstract available

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Bradykinin / analogs & derivatives*
  • Bradykinin / antagonists & inhibitors
  • Bradykinin / chemical synthesis
  • Bradykinin / metabolism
  • Bradykinin / pharmacology
  • Chelating Agents / chemical synthesis
  • Chelating Agents / metabolism
  • Chelating Agents / pharmacology
  • Ethylamines / chemical synthesis
  • Ethylamines / metabolism
  • Ethylamines / pharmacology
  • Guinea Pigs
  • Isotope Labeling / methods
  • Molecular Sequence Data
  • Organotechnetium Compounds / chemical synthesis*
  • Organotechnetium Compounds / metabolism
  • Organotechnetium Compounds / pharmacology*
  • Radionuclide Imaging
  • Receptor, Bradykinin B2
  • Receptors, Bradykinin / analysis*
  • Receptors, Bradykinin / metabolism
  • Tissue Distribution

Substances

  • Chelating Agents
  • Ethylamines
  • Organotechnetium Compounds
  • Receptor, Bradykinin B2
  • Receptors, Bradykinin
  • 2-(4-chlorophenylthio)triethylamine
  • icatibant
  • Bradykinin