The use of gene-manipulated mice in the validation of receptor binding radiotracer

Nucl Med Biol. 2003 Nov;30(8):851-60. doi: 10.1016/s0969-8051(03)00123-9.
No abstract available

Publication types

  • Comparative Study
  • Review

MeSH terms

  • Animals
  • Disease Models, Animal
  • Drug Evaluation, Preclinical / methods*
  • Gas Chromatography-Mass Spectrometry / methods*
  • Mice
  • Mice, Knockout
  • Models, Animal
  • Phenotype
  • Protein Binding
  • Radioisotope Dilution Technique*
  • Radioisotopes / pharmacokinetics*
  • Radioligand Assay / methods*
  • Radiopharmaceuticals / pharmacokinetics
  • Receptors, Cell Surface / genetics
  • Receptors, Cell Surface / metabolism*
  • Receptors, Drug / metabolism
  • Reproducibility of Results
  • Structure-Activity Relationship
  • Tomography, Emission-Computed / methods

Substances

  • Radioisotopes
  • Radiopharmaceuticals
  • Receptors, Cell Surface
  • Receptors, Drug