In vivo imaging of rat brain A1 adenosine receptor occupancy by caffeine

Eur J Nucl Med Mol Imaging. 2003 Oct;30(10):1440. doi: 10.1007/s00259-003-1273-3. Epub 2003 Aug 28.
No abstract available

Publication types

  • Comparative Study

MeSH terms

  • Adenosine A1 Receptor Antagonists*
  • Animals
  • Brain / diagnostic imaging*
  • Brain / drug effects
  • Brain / metabolism*
  • Caffeine / pharmacology*
  • Radiopharmaceuticals / pharmacokinetics
  • Rats
  • Receptor, Adenosine A1 / metabolism*
  • Reference Values
  • Tomography, Emission-Computed / methods*
  • Xanthines / pharmacokinetics*

Substances

  • 8-cyclopenta-3-(3-fluoropropyl)-1-propylxanthine
  • Adenosine A1 Receptor Antagonists
  • Radiopharmaceuticals
  • Receptor, Adenosine A1
  • Xanthines
  • Caffeine