Reversal of multidrug resistance with LY335979: functional analysis of P-glycoprotein-mediated transport activity and its modulation in vivo

J Clin Pharmacol. 2001 Jul;41(S7):29S-38S.
No abstract available

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / genetics
  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / metabolism*
  • Animals
  • Biological Transport, Active / drug effects
  • Dibenzocycloheptenes / pharmacology*
  • Drug Resistance, Multiple
  • Genes, MDR / drug effects
  • Genes, MDR / genetics*
  • Humans
  • Quinolines / pharmacology*
  • Radiopharmaceuticals
  • Technetium Tc 99m Sestamibi

Substances

  • ATP Binding Cassette Transporter, Subfamily B, Member 1
  • Dibenzocycloheptenes
  • Quinolines
  • Radiopharmaceuticals
  • zosuquidar trihydrochloride
  • Technetium Tc 99m Sestamibi