TABLE 1

In Vitro Dosimetry

ParameterIMR-05NLF
Mean D50 ± SEM (Gy)
 125I-KX10.18 ± 0.012.0 ± 0.1
 131I-KX10.35 ± 0.013.5 ± 0.3
 125I-MIBG1.1 ± 0.13.7 ± 0.3
 211At-MM40.051 ± 0.0020.56 ± 0.07
 211At-NaAtx0.20 ± 0.011.0 ± 0.1
 External γ0.71 ± 0.023.7 ± 0.1
RBE for nontargeted therapy
125I-MIBG vs. γ0.651.0
211At-NaAtx vs. γ3.63.7
211At-NaAtx vs. 125I-MIBG5.53.7
RBE for targeted therapy
125I-KX1 vs. 131I-KX11.91.8
211At-MM4 vs. 131I-KX16.76.3
211At-MM4 vs. 125I-KX13.53.6