TABLE 2
IC50 as Calculated from Competition Assays Against
125
I-Tyr
12
-Gastrin-I
Peptide analog
IC50 (nM)
DOTA-MGS5
0.4 ± 0.2
nat
In-DOTA-MGS5
0.2 ± 0.04
nat
Ga-DOTA-MGS5
0.6 ± 0.2
nat
Lu-DOTA-MGS5
0.6 ± 0.1
CP04
0.4 ± 0.1
DOTA-MG11
0.9 ± 0.3
Pentagastrin
1.0 ± 0.2