TABLE 2

IC50 as Calculated from Competition Assays Against 125I-Tyr12-Gastrin-I

Peptide analogIC50 (nM)
DOTA-MGS50.4 ± 0.2
natIn-DOTA-MGS50.2 ± 0.04
natGa-DOTA-MGS50.6 ± 0.2
natLu-DOTA-MGS50.6 ± 0.1
CP040.4 ± 0.1
DOTA-MG110.9 ± 0.3
Pentagastrin1.0 ± 0.2