TABLE 1

AUCs in Tumor, Blood, and Kidney

Parameter177Lu-RPS-063*177Lu-RPS-071177Lu-RPS-072177Lu-RPS-077
Tumor1,796 ± 76552 ± 362,747 ± 1452,266 ± 306
Blood22 ± 143 ± 14420 ± 161,018 ± 42
Kidney4,676 ± 14414 ± 13585 ± 182,114 ± 85
Tumor-to-blood82 ± 52184 ± 8596.5 ± 0.42.2 ± 0.3
Tumor-to-kidney0.4 ± 0.021.3 ± 0.094.7 ± 0.31.1 ± 0.2
  • * Data derived from previously reported results (10).

  • Data are %ID/g per hour. Tumor-to-blood and tumor-to-kidney ratios are derived from corresponding AUCs.