TABLE 1

¹⁸F-BMS-986192 In Vitro Autoradiography

		+ BMS-986192 blocking
Tissue	Total binding	0.025 nM	0.25 nM	2.5 nM	25 nM	+ Sham, 25 nM
HT29	3.59	3.67	3.94	4.02	4.14	3.40
L2987	9.58	7.16	6.04	4.21	4.92	8.92
Hu1027A^*	230.79	210.01	191.72	12.03	12.63	182.07
Hu1059A^*	89.43	72.17	50.83	10.09	5.23	86.46
Hu1063A^*	40.99	41.75	26.18	10.12	10.36	33.24
Hu1054A^*	55.96	49.89	32.39	9.28	4.20	67.11
Hu1023A^*	42.78	30.80	21.89	6.76	4.52	40.72
Hu1026A^*	21.35	17.96	11.32	5.46	4.85	24.59

↵* Denotes human NSCLC tumor sample.
All values reported as mean PSL/mm².