TABLE 1

MA1-Derived Regional VT Values for 18F-LY2459989 in Monkey Brain

VT (mL·cm−3) in brain region:
StudyGlobus pallidusCingulate cortexInsulaCaudatePutamenFrontal cortexTemporal cortexThalamusCerebellum
Baseline (n = 4)13.61 ± 2.6311.66 ± 2.949.85 ± 2.109.43 ± 2.279.05 ± 1.787.80 ± 1.887.05 ± 1.396.76 ± 1.184.62 ± 0.94
Blocking (n = 1)4.123.393.303.583.623.113.053.563.16
  • Data are reported as mean or as mean ± SD.