TABLE 1

In Vivo Biodistribution of 18F-FP-QD-RGD-BBN in Normal Mice

Organ5 min30 min60 min120 min
Blood4.57 ± 0.963.01 ± 0.501.81 ± 0.111.73 ± 0.17
Brain1.89 ± 0.331.86 ± 0.201.17 ± 0.071.04 ± 0.13
Heart2.51 ± 0.441.98 ± 0.121.39 ± 0.251.36 ± 0.30
Lung6.87 ± 2.563.49 ± 0.742.22 ± 0.421.50 ± 0.36
Liver7.03 ± 0.693.46 ± 0.842.19 ± 0.141.98 ± 0.38
Spleen1.83 ± 0.631.62 ± 0.331.04 ± 0.200.81 ± 0.15
Pancreas2.73 ± 0.771.59 ± 0.430.88 ± 0.220.61 ± 0.14
Kidneys10.8 ± 3.827.35 ± 1.692.60 ± 0.441.98 ± 0.34
Intestine2.56 ± 0.633.53 ± 0.691.94 ± 0.561.56 ± 0.28
Muscle2.20 ± 0.711.51 ± 0.380.97 ± 0.090.69 ± 0.15
Stomach2.49 ± 0.681.61 ± 0.660.96 ± 0.240.88 ± 0.10
Bone1.78 ± 0.611.72 ± 0.251.04 ± 0.240.92 ± 0.14
  • Data are average percentage injected dose per gram, mean ± SD (n = 4).