TABLE 1
PSMA Inhibitory Activities
Compound
K
i
(nM)
95% confidence interval of
K
i
4
0.41
0.34–0.56
89
Y-
4
0.36
0.2–0.51
5
3.12
1.7–5.60
89
Y-
5
0.10
0.04–0.32
6
1.80
0.83–3.92
89
Y-
6
2.99
1.91–4.69
ZJ43
1.16
0.08–2.26