Biodistribution of 86Y-4 in Mice (%ID/g)
Tissue | 1 h | 2 h | 5 h | 24 h |
Blood | 0.5 ± 0.2 | 0.1 ± 0.1 | 0.0 ± 0.0 | 0.0 ± 0.0 |
Heart | 0.3 ± 0.1 | 0.1 ± 0.0 | 0.0 ± 0.0 | 0.0 ± 0.0 |
Lung | 1.1 ± 0.2 | 0.3 ± 0.1 | 0.1 ± 0.0 | 0.0 ± 0.0 |
Liver | 0.2 ± 0.1 | 0.1 ± 0.0 | 0.1 ± 0.0 | 0.0 ± 0.0 |
Spleen | 5.1 ± 1.4 | 1.3 ± 0.5 | 0.2 ± 0.1 | 0.0 ± 0.0 |
Kidney | 245.0 ± 9.0 | 123.0 ± 48 | 23.0 ± 9.7 | 1.5 ± 0.7 |
Muscle | 0.5 ± 0.4 | 0.1 ± 0.1 | 0.1 ± 0.1 | 0.0 ± 0.0 |
Small intestines | 0.2 ± 0.0 | 0.1 ± 0.0 | 0.0 ± 0.0 | 0.0 ± 0.0 |
Large intestines | 0.3 ± 0.1 | 0.1 ± 0.0 | 0.1 ± 0.0 | 0.0 ± 0.0 |
Bladder | 1.5 ± 0.8 | 12.6 ± 12.5 | 3.6 ± 1. | 0.2 ± 0.2 |
PC-3 PIP | 29.0 ± 8.7 | 21.6 ± 3.6 | 15.7 ± 1.7 | 5.9 ± 0.8 |
PC-3 flu | 0.3 ± 0.1 | 0.1 ± 0.0 | 0.1 ± 0.0 | 0.0 ± 0.0 |
PIP to flu | 89 | 164 | 156 | 229 |
PIP to blood | 55 | 198 | 624 | 2,352 |
PIP to muscle | 54 | 140 | 191 | 1,046 |