TABLE 2

Binding Affinity of 64Cu-CB-TE1A1P-PEG4-LLP2A, 64Cu-NODAGA-PEG4-LLP2A, and Gallium-NODAGA-PEG4-LLP2A

ProbeKd (nM)Bmax (fmol/mg)
64Cu-CBTE1A1P-PEG4-LLP2A0.28 ± 0.03296 ± 4.5
64Cu-NODAGA-PEG4-LLP2A0.23 ± 0.03243 ± 5.1
IC50 (nM)Ki (nM)
Gallium-NODAGA-PEG4-LLP2A0.670.11
  • n = 3; values are expressed as mean ± SE.