TABLE 2

Tumor-to-Organ Ratios for CC49-TCO–Pretargeted 177Lu-Tetrazine 2 in Mice Bearing LS174T Colon Carcinoma Xenografts

Organ1 h3 h6 h1 d2 d4 d7 d
Blood13 ± 6196 ± 13206 ± 75307 ± 90410 ± 270446 ± 82540 ± 169*
Liver17 ± 631 ± 330 ± 930 ± 830 ± 1814 ± 48 ± 1
Kidney2 ± 13 ± 04 ± 14 ± 17 ± 36 ± 26 ± 2
Bladder3 ± 28 ± 425 ± 1020 ± 733 ± 1615 ± 37 ± 2
Muscle31 ± 18141 ± 67245 ± 108257 ± 75229 ± 145203 ± 100255 ± 152
Bone23 ± 20*95 ± 86162 ± 46159 ± 69149 ± 78114 ± 6176 ± 25
  • * n = 3.

  • Data are mean ± SD (n = 4).