TABLE 1

Peptidic Sequence, Radiochemical Purity, and Urinary Stability of 99mTc-B2702p1-20 Peptides

TracerPeptidic sequenceRCP (%)Stability (%)
99mTc-B2702pH2N-HGR ENL RIA LRY-COOH9093
99mTc-B2702p1H2N-HGR ANL RIL ARY-COOH9294
99mTc-B2702p1 mismatchH2N- HGL RAY IRA RNL-COOH9089
99mTc-B2702p2H2N-HGR ENL AIL ARY-COOH9596
99mTc-B2702p3H2N-HGR ENL RIL ARA-COOH9783
99mTc-B2702p4H2N-HGR ENL RIL AAY-COOH9592
99mTc-B2702p5H2N-HGR ENL RIL ARY-COOH50N/D
99mTc-B2702p6H2N-HGR ENA RIL ARY-COOH9395
99mTc-B2702p7H2N-HGA ENL RIL ARY-COOH9550
99mTc-B2702p8H2N-HGR ENL RIA ARY-COOH8084
99mTc-B2702p9H2N-HGR EAL RIL ARY-COOH9597
99mTc-B2702p10H2N-HGR ENL RIL ARY-COOH9599
99mTc-B2702p11H2N-HGA ENL RIA LRY-COOH9782
99mTc-B2702p12H2N-HGR ANL RIA LRY-COOH8880
99mTc-B2702p13H2N-HGR EAL RIA LRY-COOH9679
99mTc-B2702p14H2N-HGR ENA RIA LRY-COOH9676
99mTc-B2702p15H2N-HGR ENL AIA LRY-COOH9685
99mTc-B2702p16H2N-HGR ENL RAA LRY-COOH9170
99mTc-B2702p17H2N-HGR ENL RIA LAY-COOH9080
99mTc-B2702p18H2N-HGR ENL RIA LRA-COOH8881
99mTc-B2702p19H2N-HGR ANL RIL ARA-COOH8879
99mTc-B2702p20H2N-HGR ANL RIL AAY-COOH9278
  • N/D = not determined; RCP = radiochemical purity.