TABLE 2

Radiation Dosimetry Estimates per Unit Administered Activity for 18F-RGD-K5 for Human Adult Male Phantom in 1- and 4.8-Hour Bladder-Voiding Models, Based on Human Biodistribution Data

Organ1-h void model(μGy/MBq)4.8-h void model(μGy/MBq)
Urinary bladder wall103 ± 4376 ± 19
Gallbladder wall103 ± 58104 ± 59
Kidneys45 ± 1045 ± 10
Uterus14 ± 0.331 ± 1
Lower large intestine wall19 ± 527 ± 5
Liver25 ± 526 ± 5
Upper large intestine wall22 ± 1825 ± 17
Small intestine17 ± 220 ± 2
Ovaries11 ± 119 ± 0.5
Testes7.5 ± 0.413 ± 0.1
Pancreas10 ± 110 ± 1
Osteogenic cells10 ± 110 ± 1
Adrenals10 ± 110 ± 1
Muscle7 ± 0.49 ± 0.3
Stomach wall8.2 ± 18.6 ± 0.5
Red marrow6.9 ± 0.48.2 ± 0.3
Spleen7.9 ± 0.38.2 ± 0.3
Heart wall7.4 ± 0.47.5 ± 0.4
Lungs6.6 ± 0.46.6 ± 0.4
Thymus6.1 ± 0.46.2 ± 0.4
Thyroid5.9 ± 0.55.9 ± 0.5
Skin5 ± 0.35.7 ± 0.3
Breasts5.1 ± 0.35.2 ± 0.3
Total body7.8 ± 0.49.6 ± 0.3
Effective dose (μSv/MBq)15 ± 131 ± 1
  • Data are mean ± SD; n = 4.