sst1–sst5 Affinity Profile of 2 Somatostatin Analogs, Compared with SRIF-28 as Reference
| Compound | sst1 | sst2 | sst3 | sst4 | sst5 |
| SRIF-28, reference | 3.2 ± 0.4 (7) | 2.4 ± 0.2 (7) | 4.0 ± 1.1 (7) | 2.3 ± 0.5 (7) | 2.3 ± 0.3 (7) |
| DOTATATE, agonist | >1,000 (3) | 1.5 ± 0.4 (3) | >1,000 (3) | 453 ± 179 (3) | 547 ± 160 (3) |
| DOTA-BASS, antagonist | >1,000 (4) | 1.5 ± 0.4 (4) | >1,000 (4) | 287 ± 27 (4) | >1,000 (4) |
Data are expressed as 50% inhibitory concentration in nM (mean ± SEM).
Number of experiments are in parentheses.