TABLE 1

IC50 of Selected CXCR4 Ligands for Binding of 125I-FC131 to CXCR4-Expressing Jurkat Cells

CompoundIC50 (nM)
FC1314.43 ± 0.82
CPCR4-2177
natGa-CPCR4-24.99 ± 0.72
  • Data are mean ± SD of 3 experiments, except for values greater than 80 nM.