TABLE 2

Tumor-to-Tissue Ratios for 64Cu-AMD3465 for Subcutaneous Brain Tumor Xenografts

Time (min)
Ratio306090240600
U87-stb-CXCR4 to U8732.57 ± 5.5140.19 ± 7.5321.62 ± 4.3612.85 ± 4.035.38 ± 2.97
U87-stb-CXCR4 to muscle193.82 ± 108.55297.78 ± 93.83362.56 ± 153.51222.95 ± 27.62151.00 ± 29.91
U87 to muscle5.88 ± 2.937.31 ± 1.5917.53 ± 7.6418.91 ± 7.2542.04 ± 35.98
U87-stb-CXCR4 to blood56.10 ± 7.93114.76 ± 23.09138.78 ± 30.8783.47 ± 4.6327.80 ± 9.93
U87 to blood1.73 ± 0.092.85 ± 0.106.41 ± 0.636.97 ± 2.0110.04 ± 2.95