TABLE 1

Kd and Bmax Values for natGa-DOTATOC Binding to hSSTr2 Expressed by Transduced Cells

ParameterJurkat-hSSTr2 (n = 4)CHO-hSSTr2 (n = 7)U87-hSSTr2 (n = 3)C6-hSSTr2 (n = 3)
Bmax (105 sites/cell)0.36 ± 0.043.09 ± 0.402.82 ± 0.3712.5 ± 1.4
Kd (nM)5.26 ± 2.735.06 ± 0.916.90 ± 1.537.64 ± 1.43