Kd and Bmax Values for natGa-DOTATOC Binding to hSSTr2 Expressed by Transduced Cells
Parameter | Jurkat-hSSTr2 (n = 4) | CHO-hSSTr2 (n = 7) | U87-hSSTr2 (n = 3) | C6-hSSTr2 (n = 3) |
Bmax (105 sites/cell) | 0.36 ± 0.04 | 3.09 ± 0.40 | 2.82 ± 0.37 | 12.5 ± 1.4 |
Kd (nM) | 5.26 ± 2.73 | 5.06 ± 0.91 | 6.90 ± 1.53 | 7.64 ± 1.43 |