TABLE 1.

Biodistribution of 111In-R1507 and 89Zr-R1507 in Mice with Subcutaneous SUM149 Xenografts at 7 Days After Injection

Tissue111In-R1507 (%ID/g)89Zr-R1507 (%ID/g)
Blood5.6 ± 0.55.7 ± 0.7
Muscle0.7 ± 0.10.7 ± 0.1
Tumor20.9 ± 2.422.3 ± 2.5
Lung4.5 ± 0.74.6 ± 0.5
Spleen5.4 ± 0.95.7 ± 0.7
Kidney4.4 ± 0.44.9 ± 0.7
Liver2.9 ± 0.44.6 ± 0.4
Small intestine2.5 ± 0.42.5 ± 0.4
Pancreas1.0 ± 0.11.1 ± 0.1
Bone1.3 ± 0.48.2 ± 4.2
Tumor-to-liver ratio7.5 ± 1.24.8 ± 0.2
Tumor-to-blood ratio3.8 ± 0.73.9 ± 0.5
  • Values are mean ± SD.