TABLE 1

Biodistribution Results in Healthy Human Volunteers*

Time after injection (min)
Organ530602401,440
Heart
 Rest1.67 ± 0.131.55 ± 0.091.52 ± 0.061.34 ± 0.090.50 ± 0.02
 Exercise2.07 ± 0.222.01 ± 0.011.89 ± 0.041.54 ± 0.090.68 ± 0.05
Lung
 Rest1.16 ± 0.071.11 ± 0.081.04 ± 0.090.49 ± 0.120.26 ± 0.09
 Exercise1.12 ± 0.211.06 ± 0.280.91 ± 0.400.39 ± 0.070.15 ± 0.05
Liver
 Rest10.85 ± 1.726.52 ± 1.414.31 ± 1.192.85 ± 0.620.36 ± 0.16
 Exercise6.35 ± 1.273.93 ± 0.982.96 ± 0.761.89 ± 0.330.29 ± 0.08
Gallbladder
 Rest3.93 ± 1.364.15 ± 1.685.09 ± 2.374.98 ± 3.061.61 ± 1.12
 Exercise3.38 ± 0.814.05 ± 1.134.27 ± 1.704.16 ± 1.001.47 ± 0.82
Kidney
 Rest5.06 ± 1.664.25 ± 1.194.92 ± 1.873.84 ± 0.780.99 ± 0.20
 Exercise5.76 ± 0.804.91 ± 0.504.80 ± 0.814.16 ± 0.411.15 ± 0.14
Salivary glands
 Rest0.22 ± 0.020.20 ± 0.030.20 ± 0.030.17 ± 0.040.10 ± 0.03
 Exercise0.20 ± 0.050.18 ± 0.040.17 ± 0.030.13 ± 0.020.10 ± 0.03
Thyroid
 Rest0.64 ± 0.120.54 ± 0.100.53 ± 0.120.42 ± 0.070.17 ± 0.04
 Exercise0.52 ± 0.120.43 ± 0.110.44 ± 0.130.35 ± 0.090.20 ± 0.06
Spleen
 Rest0.80 ± 0.320.60 ± 0.220.48 ± 0.110.32 ± 0.060.17 ± 0.04
 Exercise0.76 ± 0.230.61 ± 0.160.54 ± 0.180.42 ± 0.130.19 ± 0.10
  • * Data are percentage injected activity per organ.