Time after injection (min) | ||||
---|---|---|---|---|
Region | 2 | 30 | 60 | 120 |
Blood | 0.26 ± 0.03 | 0.23 ± 0.06 | 0.18 ± 0.02 | 0.12 ± 0.03 |
Heart | 0.71 ± 0.07 | 0.41 ± 0.03 | 0.30 ± 0.10 | 0.22 ± 0.01 |
Muscle | 0.14 ± 0.03 | 0.17 ± 0.02 | 0.13 ± 0.01 | 0.10 ± 0.01 |
Lung | 0.94 ± 0.04 | 0.69 ± 0.03 | 0.54 ± 0.14 | 0.35 ± 0.03 |
Kidney | 2.10 ± 0.17 | 1.06 ± 0.06 | 0.84 ± 0.09 | 0.55 ± 0.06 |
Pancreas | 2.51 ± 0.22 | 5.50 ± 0.97 | 4.98 ± 0.24 | 2.76 ± 0.61 |
Spleen | 1.46 ± 0.15 | 1.03 ± 0.18 | 0.83 ± 0.18 | 0.48 ± 0.04 |
Liver | 3.53 ± 0.56 | 2.82 ± 0.24 | 2.47 ± 0.30 | 1.47 ± 0.13 |
Skin | 0.23 ± 0.05 | 0.28 ± 0.01 | 0.23 ± 0.04 | 0.16 ± 0.02 |
Whole brain | 0.71 ± 0.05 | 0.62 ± 0.08 | 0.42 ± 0.04 | 0.35 ± 0.02 |
Regional brain | ||||
Cerebellum | 0.63 ± 0.03 | 0.40 ± 0.04 | 0.28 ± 0.04 | 0.20 ± 0.01 |
Striatum | 1.52 ± 0.20 | 2.25 ± 0.48 | 1.85 ± 0.26 | 1.42 ± 0.54 |
Hippocampus | 0.68 ± 0.07 | 0.61 ± 0.12 | 0.36 ± 0.08 | 0.23 ± 0.03 |
Cortex | 0.65 ± 0.02 | 0.44 ± 0.06 | 0.27 ± 0.07 | 0.20 ± 0.06 |
Remainder | 0.70 ± 0.04 | 0.62 ± 0.08 | 0.44 ± 0.08 | 0.36 ± 0.08 |
Hypothalamus | 1.23 ± 0.29 | 1.46 ± 0.40 | 1.21 ± 0.20 | 0.83 ± 0.10 |
Data are % dose/g, average of 3 rats ± SD. Regional brain distribution data are % dose/g ± SD.