TABLE 1

Biodistribution of 18F-BMS-747158-02 in Male Wistar Rats

Mean (SD) %ID/g at following time after injection*:
Tissue10 min60 min
Blood0.12 (0.01)0.15 (0.01)
Lungs0.32 (0.08)0.21 (0.02)
Heart3.07 (0.66)2.06 (0.83)
Liver0.99 (0.23)0.38 (0.05)
Stomach0.74 (0.42)0.38 (0.07)
Spleen0.20 (0.01)0.15 (0.01)
Pancreas1.01 (0.19)0.36 (0.08)
Intestines0.45 (0.06)0.29 (0.01)
Kidneys2.00 (0.42)0.62 (0.04)
Adrenal glands0.20 (0.04)0.21 (0.05)
Bone0.17 (0.03)0.20 (0.01)
Brain1.07 (0.28)0.58 (0.08)
Muscle0.17 (0.03)0.20 (0.03)
  • * n = 3 per time point.