TABLE 3

Tissue Distribution (%ID/g) of 64Cu-TP3939 in PC3 Tumor-Bearing Nude Mice (n = 5)

Tissue4 h24 hP
Muscle1.94 ± 0.851.15 ± 0.180.17
Intestine11.00 ± 1.647.67 ± 2.480.06
Heart9.13 ± 5.634.14 ± 0.650.19
Lungs34.31 ± 9.7619.93 ± 5.560.06
Blood3.85 ± 1.142.38 ± 0.260.07
Spleen19.22 ± 9.133.56 ± 0.380.03
Kidneys18.38 ± 9.9510.06 ± 0.420.21
Liver55.00 ± 12.6227.58 ± 2.180.01
Tumor7.48 ± 3.635.78 ± 0.660.47
T/M ratio3.98 ± 1.435.17 ± 1.320.29
T/B ratio1.94 ± 0.662.46 ± 0.450.28