Receptor Binding Affinity Measurements on Selected Peptides Using 125I-G17 as Radioligand
| Peptide | EC50/Ki (nM) |
|---|---|
| DOTA-CCK8 | 3.1/2.1 |
| DOTA-H6-Met | 3.1/2.1 |
| DOTA-H2-Met | 5.7/3.9 |
| DOTA-H2-Met(O) | 1,300.0/900.0 |
| DOTA-H6-Nle | 5.7/3.8 |
| DOTA-H2-Nle | 16.7/11.3 |
| MG0 | 2.5/1.7 |
| MG11 | 3.4/2.4 |