Injection 1 (T = 0 min) | Injection 2 | Injection 3 | ||||||||
---|---|---|---|---|---|---|---|---|---|---|
Subject no. | Modality/protocol | Duration (min) | SA* (GBq/μmol) | J1* (mg) | Time (min) | J2* (mg) | J2 (mg) | Time (min) | J3* (mg) | J3 (mg) |
1 | SPECT/1 | 160 | 156.81 | 0.133 | 70 | — | 0.73 | 110 | 0.140 | 1.46 |
2 | SPECT/1 | 160 | 156.18 | 0.138 | 70 | — | 1.28 | 110 | 0.154 | 1.28 |
3 | SPECT/1 | 160 | 95.68 | 0.212 | 70 | — | 1.34 | 110 | 0.248 | 1.34 |
4 | SPECT/1 | 160 | 91.69 | 0.219 | 70 | — | 2.00 | 110 | 0.322 | 2.00 |
5 | SPECT/2 | 160 | 68.78 | 0.335 | 70 | 0.381 | 1.64 | 110 | — | 1.64 |
6 | SPECT/2 | 160 | 113.18 | 0.201 | 70 | 0.229 | 1.44 | 110 | — | 1.44 |
7 | SPECT/2 | 160 | 107.41 | 0.218 | 70 | 0.238 | 1.44 | 110 | — | 1.44 |
8 | SPECT/2 | 160 | 100.86 | 0.232 | 70 | 0.252 | 1.54 | 110 | — | 1.54 |
7 | PET | 104 | 109.96 | 0.467 | 30 | — | 0.70 | 60 | 3.490 | 1.40 |
↵* Specific activity at beginning of experiment.
Doses Ji* and Ji correspond, respectively, to labeled and unlabeled ligand doses injected during the ith injection.