TABLE 1

Selected Receptor Tracers

TracerAbbreviationTarget
11C-Cocaine, 11C-methylphenidateDAT
11C-NomifensineDAT
11C-WIN-35428, 11C-PE2IDAT
18F-2β-Carbomethoxy-3β-(4-fluorophenyl)tropaneCFTDAT
11C-DihydrotetrabenazineDTBZVMAT2
11C-SCH-23390D1
11C-N-MethylspiperoneNMSPD2, 5-HT2
18F-N-Methylspiperone
18F-FluoroethylspiperoneFESPD2, 5-HT2
11C-RacloprideRACD2
18F-FallyprideD2
N-1-11C-PropylnorapomorphineD2 (agonist)
11C-l-DeprenylMAO-A
11C-N-Methyl-4-piperidylbenzilateNMPBMuscarinic receptors
N-11C-Methylpiperdin-4-yl-propionateMP4P, PMPAChE
N-11C-Methyl-4-piperidyl-acetateMP4A, AMPAChE
11C(+)-McN56525-HTT
11C-3-Amino-4-(2-dimethylaminomethyl-phenylsulfanyl)benzonitrileDASB5-HTT
11C-WAY-100635WAY5-HT1A receptor
18F-Altanserin5-HT2A receptor
11C-FlumazenilFMZGABAA/benzodiazepine receptors
11C-PK-11195PKPeripheral benzodiazepine receptors
11C-CarfentanylOpioid μ receptor
11C-DiprenorphineDPNOpioid receptors
18F-CyclofoxyOpioid receptors
18F-CPFPX, 11C-MPDXAdenosine A1 receptor
  • DAT = dopamine transporter; VMAT2 equals vesicular monoamine transporter type 2; D1 equals dopamine 1 receptor; D2 equals dopamine 2 receptor; 5-HT equals 5-hydroxytryptamine (serotonin) receptor; 5-HTT equals 5-hydroxytryptamine (serotonin) transporter; MAO-A equals monoamino-oxidase A; AChE equals acetylcholinesterase; GABA equals γ-aminobutyric acid receptor.