TABLE 1

Biodistribution Data of 64Cu-TETA-SCK-Folate in KB Tumor Cell Xenograft-Bearing Athymic Nude Female Mice (n = 4)

Biodistribution%ID/g%ID/organ
10 min1 h4 h24 h10 min1 h4 h24 h
Blood2.1 ± 0.22.1 ± 0.22.5 ± 0.32.6 ± 0.63.1 ± 0.23.4 ± 0.24.2 ± 0.34.3 ± 0.9
Lung39.7 ± 5.110.9 ± 3.814.4 ± 5.910.8 ± 1.45.1 ± 0.91.5 ± 0.22.1 ± 0.91.5 ± 0.2
Liver56.0 ± 7.138.4 ± 7.933.8 ± 2.621.5 ± 2.952.3 ± 5.641.7 ± 3.034.1 ± 2.525.2 ± 2.9
Spleen18.3 ± 6.310.8 ± 3.28.8 ± 0.54.7 ± 1.01.5 ± 0.41.0 ± 0.30.8 ± 0.20.5 ± 0.2
Kidney7.2 ± 1.68.1 ± 1.87.9 ± 0.88.5 ± 1.31.2 ± 0.31.3 ± 0.21.4 ± 0.21.5 ± 0.4
Muscle0.8 ± 0.10.8 ± 0.20.9 ± 0.21.0 ± 0.17.2 ± 0.57.5 ± 1.38.6 ± 1.79.5 ± 1.3
Heart2.3 ± 0.22.7 ± 0.53.7 ± 0.34.3 ± 0.50.2 ± 0.00.3 ± 0.10.4 ± 0.00.5 ± 0.0
Tumor3.4 ± 1.22.3 ± 0.75.9 ± 2.82.9 ± 3.10.04 ± 0.020.12 ± 0.020.04 ± 0.020.09 ± 0.07
  • Data are presented as percentage injected dose per gram (%ID/g) and percentage injected dose per organ (%ID/organ) ± SD.