TABLE 1

PET-Determined FK506 Concentrations After 0.1 mg/kg Intravenous Administration of 11C-FK506 to Anesthetized Monkeys

Time (min)Cortex (ng/g)Striatum (ng/g)Whole blood (ng/mL)
520.0 ± 2.113.4 ± 1.5205.8 ± 9.3
1520.0 ± 1.714.1 ± 1.7147.6 ± 12.8
  • Data are mean ± SD for 3 animals.