TABLE 3

%ID/g Determined by Whole-Body Autoradiography or Tissue Dissection

TissueBiodistribution methodn1 h3 h6 h16 h24 h
SpleenAutoradiography236.0039.2033.7012.304.77
Tissue dissection339.1034.4028.5010.406.25
Mean537.8036.3030.6011.205.66
Lymph nodeAutoradiography29.3017.4013.604.162.51
Tissue dissection39.2020.1017.403.943.11
Mean59.2419.0015.904.032.87
StomachAutoradiography27.9916.6014.201.871.33
Tissue dissection37.0710.8021.502.620.61
Mean57.4413.1018.602.320.90
LungAutoradiography214.509.064.420.250.15
Tissue dissection317.007.703.890.350.17
Mean516.008.244.110.310.16
DuodenumAutoradiography23.455.675.950.570.38
Tissue dissection35.184.524.801.680.37
Mean54.494.985.260.640.38
HeartAutoradiography29.286.923.560.140.12
Tissue dissection37.493.722.030.150.07
Mean58.215.002.640.150.09
KidneyAutoradiography25.644.933.030.260.17
Tissue dissection35.562.962.290.210.09
Mean55.593.752.590.220.13
LiverAutoradiography26.826.223.070.260.15
Tissue dissection34.372.351.740.170.08
Mean55.353.902.270.210.11
MuscleAutoradiography21.001.130.880.070.03
Tissue dissection31.531.731.120.060.06
Mean51.321.481.020.060.05
PancreasAutoradiography22.403.202.750.220.16
OvaryAutoradiography26.835.212.150.230.18
Bone marrowAutoradiography26.617.053.990.700.34
ThymusAutoradiography23.232.751.370.410.18
UterusAutoradiography24.067.703.020.220.18
ThyroidAutoradiography231.5032.20157.0075.70229.00
FemurTissue dissection33.212.532.070.310.11
Whole bodyAutoradiography23.294.443.010.400.33