Selectivity of Ligands for Monoamine Transporters (Ki, nmol/L)
Ligand | SERT | DAT | NET |
---|---|---|---|
4-F-ADAM | 0.081 ± 0.006* | 2,267 ± 188* | 117 ± 23* |
(4.8 ± 1.3)† | (5,358 ± 1,959)† | (137.2 ± 23.2)† | |
(+)McN5652 | 0.009 ± 0.002* | 112 ± 23* | 11.3 ± 3.3* |
AFM | 1.8 ± 0.3† | 2,055 ± 917† | 95.5 ± 33.8† |
ADAM | 0.013 ± 0.003* | 840 ± 100* | 699 ± 80* |
DASB | 1.10 ± 0.04‡ | 1,423 ± 103‡ | 1,350 ± 221‡ |