TABLE 1.

Biodistribution Results for 177Lu-TEFAPI-06 and 177Lu-TEFAPI-07

177Lu-TEFAPI-06177Lu-TEFAPI-07
24 h96 h24 h96 h
OrganMeanSDMeanSDMeanSDMeanSD
Blood12.321.332.250.685.641.490.510.24
Pancreas2.010.260.750.422.160.690.530.22
Spleen3.000.663.661.222.690.871.880.34
Small intestine2.550.640.610.281.190.260.160.09
Large intestine1.660.270.530.351.150.330.100.15
Liver2.980.641.740.573.210.812.310.17
Kidney3.200.842.660.548.672.3010.163.28
Stomach1.750.170.540.211.200.450.290.14
Fat1.860.901.551.171.821.180.480.25
Muscle1.090.180.450.051.000.370.280.16
Bone1.320.300.350.201.710.630.180.28
Lung4.331.441.950.702.580.750.730.28
Heart3.701.591.510.422.531.190.620.17
Brain0.370.080.090.030.230.09−0.010.04
Tumor8.680.737.332.287.872.087.572.68
  • Data are %ID/g.