Most Relevant α7 nAChR PET Tracers
Tracer name | Formula |
---|---|
11C-CHIBA-1001 | 4-11C-methylphenyl)-1,4-diazabicyclo[3.2.2]nonane-4-carboxylate |
11C-NS14492 | (2-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-5-(1-11C-methyl-1H-pyrrol-2-yl)-1,3,4-oxadiazole) |
18F-NS10743 | 2-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-5-(4-18F-fluorophenyl)-1,3,4-oxadiazole |
18F-NS14490 | (1R,5S)-3-(6-(1-(2-18F-fluoroethyl)indol-5-yl)pyridazin-3-yl)-9-methyl-3,9-diazabicyclo[3.3.1]nonane |
18F-DBT10 | 7-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-2-18F-fluorodibenzo[b,d ]thiophene 5,5-dioxide |
18F-ASEM | 7-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-4-18F-fluorodibenzo[b,d ]thiophene 5,5-dioxide |
11C-MeQAA | (1S,3R,4S)-quinuclidin-3-yl 3-(11C-methylamino)benzoate |