TABLE 3

Most Relevant α7 nAChR PET Tracers

Tracer nameFormula
11C-CHIBA-10014-11C-methylphenyl)-1,4-diazabicyclo[3.2.2]nonane-4-carboxylate
11C-NS14492(2-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-5-(1-11C-methyl-1H-pyrrol-2-yl)-1,3,4-oxadiazole)
18F-NS107432-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-5-(4-18F-fluorophenyl)-1,3,4-oxadiazole
18F-NS14490(1R,5S)-3-(6-(1-(2-18F-fluoroethyl)indol-5-yl)pyridazin-3-yl)-9-methyl-3,9-diazabicyclo[3.3.1]nonane
18F-DBT107-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-2-18F-fluorodibenzo[b,d ]thiophene 5,5-dioxide
18F-ASEM7-(1,4-diazabicyclo[3.2.2]nonan-4-yl)-4-18F-fluorodibenzo[b,d ]thiophene 5,5-dioxide
11C-MeQAA(1S,3R,4S)-quinuclidin-3-yl 3-(11C-methylamino)benzoate