TABLE 1.

PET Scan Parameters

Test–retest (n = 6)Occupancy (n = 9)
ParameterTestRetestBaselinePostdose 1Postdose 2
Injected dose (MBq)618 ± 134519 ± 196528 ± 126540 ± 132532 ± 109
Injected mass (μg)0.90 ± 0.570.75 ± 0.591.16 ± 1.131.19 ± 1.190.93 ± 0.48
Plasma free fraction47% ± 5%50% ± 7%50% ± 7%51% ± 5%52% ± 6%