TABLE 1

Biodistribution Data for (±)-11C-YJH08 Vs. (±)-18F-YJH08

Tissue(±)-11C-YJH08(±)-18F-YJH08
Blood2.25 ± 0.212.22 ± 0.14
Brain1.81 ± 0.171.93 ± 0.07
Heart4.47 ± 0.434.15 ± 0.31
Liver12.19 ± 1.2211.08 ± 0.92
Spleen2.22 ± 0.332.46 ± 0.53
Kidneys5.82 ± 0.285.79 ± 1.07
Supraspinal brown fat depot9.8 ± 2.839.01 ± 2.07
Adrenal gland13.88 ± 7.1512.19 ± 6.46
Muscle1.53 ± 0.131.53 ± 0.12
Bone1.19 ± 0.131.3 ± 0.23
  • Data are percentage injected dose per gram of tissue and were collected in intact male C57BL6/J mice at 20 min after injection. Data for (±)-18F-YJH08 were previously reported (6).