Research ArticleBasic Science Investigations
Discovery and Development of 11C-Lu AE92686 as a Radioligand for PET Imaging of Phosphodiesterase10A in the Brain
Jan Kehler, John Paul Kilburn, Sergio Estrada, Søren Rahn Christensen, Anders Wall, Alf Thibblin, Mark Lubberink, Christoffer Bundgaard, Lise Tøttrup Brennum, Björn Steiniger-Brach, Claus Tornby Christoffersen, Stine Timmermann, Mads Kreilgaard, Gunnar Antoni, Benny Bang-Andersen and Jacob Nielsen
Journal of Nuclear Medicine September 2014, 55 (9) 1513-1518; DOI: https://doi.org/10.2967/jnumed.114.140178
Jan Kehler
1Division of Discovery Chemistry and DMPK, H. Lundbeck A/S, Valby, Denmark
John Paul Kilburn
1Division of Discovery Chemistry and DMPK, H. Lundbeck A/S, Valby, Denmark
Sergio Estrada
2Preclinical PET Platform, Department of Medicinal Chemistry, Uppsala University, Uppsala, Sweden
Søren Rahn Christensen
3Department of Clinical Pharmacology, H. Lundbeck A/S, Valby, Denmark
Anders Wall
4Nuclear Medicine and PET, Uppsala University and Uppsala University Hospital, Uppsala, Sweden
Alf Thibblin
2Preclinical PET Platform, Department of Medicinal Chemistry, Uppsala University, Uppsala, Sweden
Mark Lubberink
4Nuclear Medicine and PET, Uppsala University and Uppsala University Hospital, Uppsala, Sweden
Christoffer Bundgaard
1Division of Discovery Chemistry and DMPK, H. Lundbeck A/S, Valby, Denmark
Lise Tøttrup Brennum
5Division of Synaptic Transmission, H. Lundbeck A/S, Valby, Denmark
Björn Steiniger-Brach
5Division of Synaptic Transmission, H. Lundbeck A/S, Valby, Denmark
Claus Tornby Christoffersen
6Department of Molecular Pharmacology, H. Lundbeck A/S, Valby, Denmark
Stine Timmermann
7Department of Quantitative Pharmacology, H. Lundbeck A/S, Valby, Denmark; and
Mads Kreilgaard
8Department of Drug Design and Pharmacology, University of Copenhagen, Copenhagen, Denmark
Gunnar Antoni
2Preclinical PET Platform, Department of Medicinal Chemistry, Uppsala University, Uppsala, Sweden
Benny Bang-Andersen
1Division of Discovery Chemistry and DMPK, H. Lundbeck A/S, Valby, Denmark
8Department of Drug Design and Pharmacology, University of Copenhagen, Copenhagen, Denmark
Jacob Nielsen
5Division of Synaptic Transmission, H. Lundbeck A/S, Valby, Denmark
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Journal of Nuclear Medicine
Vol. 55, Issue 9
September 1, 2014
Discovery and Development of 11C-Lu AE92686 as a Radioligand for PET Imaging of Phosphodiesterase10A in the Brain
Jan Kehler, John Paul Kilburn, Sergio Estrada, Søren Rahn Christensen, Anders Wall, Alf Thibblin, Mark Lubberink, Christoffer Bundgaard, Lise Tøttrup Brennum, Björn Steiniger-Brach, Claus Tornby Christoffersen, Stine Timmermann, Mads Kreilgaard, Gunnar Antoni, Benny Bang-Andersen, Jacob Nielsen
Journal of Nuclear Medicine Sep 2014, 55 (9) 1513-1518; DOI: 10.2967/jnumed.114.140178
Discovery and Development of 11C-Lu AE92686 as a Radioligand for PET Imaging of Phosphodiesterase10A in the Brain
Jan Kehler, John Paul Kilburn, Sergio Estrada, Søren Rahn Christensen, Anders Wall, Alf Thibblin, Mark Lubberink, Christoffer Bundgaard, Lise Tøttrup Brennum, Björn Steiniger-Brach, Claus Tornby Christoffersen, Stine Timmermann, Mads Kreilgaard, Gunnar Antoni, Benny Bang-Andersen, Jacob Nielsen
Journal of Nuclear Medicine Sep 2014, 55 (9) 1513-1518; DOI: 10.2967/jnumed.114.140178