[PDF][PDF] Preclinical evaluation of technetium-99m-labeled somatostatin receptor-binding peptides

…, BR Moyer, J Lister-James, BJ McBride… - Journal of Nuclear …, 1996 - Soc Nuclear Med
[DTPAjoctreotide. Conclusion: The high SSTR-binding affinity and high, receptor-specific
and saturable in vivo tumor uptake indicate that"" Tc-PSS? and 99mTc-P829 are promising …

Improved iodine radiolabels for monoclonal antibody therapy

…, MJ Mattes, S Chen, L Reed, G Newsome, BJ McBride… - Cancer Research, 2003 - AACR
A major disadvantage of 131 iodine (I)-labeled monoclonal antibodies (MAbs) for
radioimmunotherapyhas been the rapid diffusion of iodotyrosine from target cells afterinternalization …

Pretargeting with bispecific anti-renal cell carcinoma x anti-DTPA (In) antibody in 3 RCC models

…, AC Soede, BJ McBride… - Journal of Nuclear …, 2005 - Soc Nuclear Med
We have developed an efficient pretargeting strategy for renal cell carcinoma (RCC) based
on a biologically produced bispecific monoclonal antibody (bs-mAb). Tumor targeting with …

[PDF][PDF] Pre-clinical evaluation of technetium-99m platelet receptor-binding peptide

…, BR Moyer, DA Pearson, BJ McBride… - Journal of Nuclear …, 1997 - Soc Nuclear Med
P748 in deep vein and pulmonary thrombi was assessed in a canine thrombosis model and
the biodistribution of 99nrTc-P748was de termined in rats. Results: P748 peptide inhibited …

Labeling of Monoclonal Antibodies with Diethylenetriaminepentaacetic Acid-Appended Radioiodinated Peptides Containing d-Amino Acids

…, MJ Mattes, R Stein, BJ McBride… - Bioconjugate …, 1999 - ACS Publications
The optimal use of radioiodinated internalizing monoclonal antibodies (mAbs) for
radioimmunotherapy necessitates the development of practical methods for increasing the level of …

Epoxyannulation. 4. Reactions of 1, 5-, 1, 6-, and 1, 7-oxosulfonium salts

ME Garst, BJ McBride, AT Johnson - The Journal of Organic …, 1983 - ACS Publications
(, CH2) ni(C (CH2) n_n-i taine generation, 14 from ylide reactions with unhindered enones,
15 and from ylide reactions with 4-ieri-butylcyclo-hexanone. 15 All of these tests for …

Residualizing iodine markedly improved tumor targeting using bispecific antibody-based pretargeting

…, E Oosterwijk, JEM van Eerd, BJ McBride… - Journal of Nuclear …, 2005 - Soc Nuclear Med
Previous studies have shown that pretargeting allows rapid visualization of renal cell
carcinomas (RCC) with an 111 In-labeled bivalent peptide. For radioimmunotherapy, a β-emitting …

Cycloadditions of 4-pyrones. An approach to colchicine

BJ McBride, ME Garst - Tetrahedron, 1993 - Elsevier
The 4-pyrone, [5-acetoxy-4-oxo-4H -pyran-2-yl]carbonyl chloride was coupled with malonate
anion of bis(2,2,2-trichloroethyl) 2-ethenyl-3,4,5-trimethoxybenzylpropanedioate and …

A simple method for the preparation of 123I and 125I labeled iodobenzodiazepines

BJ McBride, RM Baldwin, JM Kerr, JL Wu - International journal of radiation …, 1991 - Elsevier
The tributyltin derivative of the benzodiazepine antagonist ethyl 7-iodo-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a]
[1,4]benzodiazepine-3-carboxylate (Ro 16-0154) was synthesized …

Synthesis, Characterization, and Crystal Structure of Neutral Rhenium (V) Complexes with S-Substituted N2S2 Ligands

…, RM Baldwin, EF Byrne, BJ McBride - Inorganic …, 1994 - ACS Publications
CH2CH= CH2 and CH2CH2-CH3, showed them to consist of a square pyramidal RevON2S2
core. ReO [CH2= CHCH2SC (CH3) 2CH2N (o-C6lLt) NCH2C (CH3) 2S], CnH25N20S2Re…