TABLE 1

Binding Affinities (Kd ± SD, nmol/L; n = 3) of NLS-Derivatives and DOTA-TOC Labeled with 111In for sstr2A

CompoundKd (sstr2A)
111In-DOTA-TOC2.48 ± 0.51
111In-(1)280 ± 140
111In-(2)15.6 ± 1.2
111In-(3)7.4 ± 1.3
111In-(4)>10,000